Compile Data Set for Download or QSAR
Found 102 of ki data for complexid = 50000268
LigandPNGBDBM50180775(CHEMBL386763 | FV-Aib-TDVGPFAF | [Aib29,Asp31,Pro3...)copy SMILEScopy InChI
Affinity DataKi:  0.00200nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280526HPubMed
LigandPNGBDBM50541408(CHEMBL4643140)copy SMILEScopy InChI
Affinity DataKi:  0.00400nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0Z1GPubMed
LigandPNGBDBM50184069(CHEMBL207197 | N-((R)-1-((S)-6-amino-1-oxo-1-(4-(p...)copy SMILEScopy InChI
Affinity DataKi:  0.00500nMAssay Description:Displacement of [125I]CGRP from human cloned CLR/RAMP1 receptor expressed in E10 cellsMore data for this Ligand-Target Pair
LigandPNGBDBM50180778(CHEMBL2371891 | FV-Hyp-TDVGPFAF)copy SMILEScopy InChI
Affinity DataKi:  0.00600nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280526HPubMed
LigandPNGBDBM50541406(CHEMBL4649325)copy SMILEScopy InChI
Affinity DataKi:  0.00700nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0Z1GPubMed
LigandPNGBDBM50385312(CHEMBL2035984)copy SMILEScopy InChI
Affinity DataKi:  0.0140nMAssay Description:Displacement of [125I]CGRP from human recombinant CALCRL/RAMP1 receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7BG1PubMed
LigandPNGBDBM362044(US10272077, Example 4 | US9833448, Example 4)copy SMILEScopy InChI
Affinity DataKi:  0.0150nMAssay Description:Antagonist activity at human CLR/RAMP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0Z1GPubMed
LigandPNGBDBM50385311(CHEMBL2035985)copy SMILEScopy InChI
Affinity DataKi:  0.0160nMAssay Description:Displacement of [125I]CGRP from human recombinant CALCRL/RAMP1 receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7BG1PubMed
LigandPNGBDBM391716(N-[(2R)-3-(7-methyl-1H- | US10300056, Example 1 | ...)copy SMILES
Affinity DataKi:  0.0200nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JKRPubMed
LigandPNGBDBM50062162(CHEMBL264010 | FVPTDVGPFAF)copy SMILEScopy InChI
Affinity DataKi:  0.0200nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280526HPubMed
LigandPNGBDBM50180781(CHEMBL2371890 | FV-Tic-TDVGPFAF)copy SMILEScopy InChI
Affinity DataKi:  0.0200nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280526HPubMed
LigandPNGBDBM50541407(CHEMBL4638635)copy SMILEScopy InChI
Affinity DataKi:  0.0200nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0Z1GPubMed
LigandPNGBDBM50356282(CHEMBL1910936)copy SMILEScopy InChI
Affinity DataKi:  0.0220nMAssay Description:Displacement of [125I]CGRP from human recombinant CALCRL/RAMP1 receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7BG1PubMed
LigandPNGBDBM50539955(CHEMBL4638938)copy SMILEScopy InChI
Affinity DataKi:  0.0251nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JKRPubMed
LigandPNGBDBM50385313(CHEMBL2035982)copy SMILEScopy InChI
Affinity DataKi:  0.0280nMAssay Description:Displacement of [125I]CGRP from human recombinant CALCRL/RAMP1 receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7BG1PubMed
LigandPNGBDBM391726(N-[(2R)-3-(7-methyl-1H- | US10300056, Example 11 |...)copy SMILES
Affinity DataKi:  0.0316nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JKRPubMed
LigandPNGBDBM50184069(CHEMBL207197 | N-((R)-1-((S)-6-amino-1-oxo-1-(4-(p...)copy SMILEScopy InChI
Affinity DataKi:  0.0316nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
LigandPNGBDBM391723(3,5-dibromo-Nalpha-{[4-(2- | US10300056, Example 8...)copy SMILES
Affinity DataKi:  0.0398nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JKRPubMed
LigandPNGBDBM50385314(CHEMBL2035981)copy SMILEScopy InChI
Affinity DataKi:  0.0400nMAssay Description:Displacement of [125I]CGRP from human recombinant CALCRL/RAMP1 receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7BG1PubMed
LigandPNGBDBM391726(N-[(2R)-3-(7-methyl-1H- | US10300056, Example 11 |...)copy SMILES
Affinity DataKi:  0.0400nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0Z1GPubMed
LigandPNGBDBM50444982(CHEMBL3099918)copy SMILEScopy InChI
Affinity DataKi:  0.0400nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50385309(CHEMBL2035983)copy SMILEScopy InChI
Affinity DataKi:  0.0470nMAssay Description:Displacement of [125I]CGRP from human recombinant CALCRL/RAMP1 receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7BG1PubMed
LigandPNGBDBM50444972(CHEMBL3099931)copy SMILEScopy InChI
Affinity DataKi:  0.0500nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM103499(US8552023, 11)copy SMILEScopy InChI
Affinity DataKi:  0.0500nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM391725(N-[(2R)-3-(7-methyl-1H- | US10300056, Example 10 |...)copy SMILES
Affinity DataKi:  0.0631nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JKRPubMed
LigandPNGBDBM361594(US10272077, Example 1 | US9833448, Example 1)copy SMILEScopy InChI
Affinity DataKi:  0.0670nMAssay Description:Antagonist activity at human CLR/RAMP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0Z1GPubMed
LigandPNGBDBM391718(N-[(2R)-3-(7-methyl-1H- | US10300056, Example 3 | ...)copy SMILES
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JKRPubMed
LigandPNGBDBM391724(3,5-dibromo-Nalpha-{[4-(2- | US10300056, Example 9...)copy SMILEScopy InChI
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JKRPubMed
LigandPNGBDBM50444980(CHEMBL3099920)copy SMILEScopy InChI
Affinity DataKi:  0.0800nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50444984(CHEMBL3099916)copy SMILEScopy InChI
Affinity DataKi:  0.0900nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50539954(CHEMBL4636143)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JKRPubMed
LigandPNGBDBM50541405(CHEMBL4633407)copy SMILEScopy InChI
Affinity DataKi:  0.110nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0Z1GPubMed
LigandPNGBDBM103501(US8552023, 13)copy SMILEScopy InChI
Affinity DataKi:  0.130nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50444971(CHEMBL3099932)copy SMILEScopy InChI
Affinity DataKi:  0.130nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50444976(CHEMBL3099926)copy SMILEScopy InChI
Affinity DataKi:  0.130nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50541410(CHEMBL4637301)copy SMILEScopy InChI
Affinity DataKi:  0.150nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0Z1GPubMed
LigandPNGBDBM50444987(CHEMBL3099939)copy SMILEScopy InChI
Affinity DataKi:  0.160nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50444975(CHEMBL3099927)copy SMILEScopy InChI
Affinity DataKi:  0.160nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50444974(CHEMBL3099929)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50444986(CHEMBL3099914)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50444981(CHEMBL3099919)copy SMILEScopy InChI
Affinity DataKi:  0.220nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50444968(CHEMBL3099935)copy SMILEScopy InChI
Affinity DataKi:  0.220nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50385310(CHEMBL2035986)copy SMILEScopy InChI
Affinity DataKi:  0.25nMAssay Description:Displacement of [125I]CGRP from human recombinant CALCRL/RAMP1 receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7BG1PubMed
LigandPNGBDBM50541413(CHEMBL4649671)copy SMILEScopy InChI
Affinity DataKi:  0.25nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0Z1GPubMed
LigandPNGBDBM50444977(CHEMBL3099924)copy SMILEScopy InChI
Affinity DataKi:  0.310nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50444988(CHEMBL3099913)copy SMILEScopy InChI
Affinity DataKi:  0.350nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM103497(US8552023, 29)copy SMILEScopy InChI
Affinity DataKi:  0.450nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50444967(CHEMBL3099936)copy SMILEScopy InChI
Affinity DataKi:  0.610nMAssay Description:Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB8393PubMed
LigandPNGBDBM50180777(CHEMBL427759 | FV((1R,2R,3R)-beta-aminocyclopropan...)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280526HPubMed
LigandPNGBDBM50224431(CHEMBL236593 | MK-0974 | N-[(3R,6S)-6-(2,3-difluor...)copy SMILEScopy InChI
Affinity DataKi:  0.770nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
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